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First report of safety, PK, and preliminary antitumor activity of the oral EGFR/HER2 exon 20 inhibitor TAK-788 (AP32788) in non–small cell lung cancer (NSCLC). |
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Stock and Other Ownership Interests - Rain Therapeutics |
Honoraria - ARIAD; AstraZeneca; Guardant Health; Pfizer; Spectrum Pharmaceuticals; Takeda; Trovagene |
Consulting or Advisory Role - AstraZeneca; GreenPeptide; Ignyta; OncoMed; Pfizer; Trovagene |
Research Funding - Ignyta (Inst) |
Patents, Royalties, Other Intellectual Property - Licensing Fees from Abbott Molecular for Patent PCT/US2013/057495; Licensing fees from Ignyta for biologic materials (Inst) |
Travel, Accommodations, Expenses - ARIAD; Guardant Health; Ignyta |
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Consulting or Advisory Role - Genentech |
Research Funding - ARIAD (Inst); GlaxoSmithKline (Inst); Infinity Pharmaceuticals (Inst); Millennium (Inst); Novartis (Inst); Pfizer (Inst); Roche/Genentech (Inst) |
Patents, Royalties, Other Intellectual Property - Patent application submitted covering pulsatile use of erlotinib to treat or prevent brain metastases (Inst) |
Travel, Accommodations, Expenses - Merck Sharp & Dohme |
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Research Funding - Abbvie (Inst); Astellas Pharma (Inst); AstraZeneca (Inst); Boehringer Ingelheim (Inst); CytomX Therapeutics (Inst); Ignyta (Inst); Incyte (Inst); LAM Therapeutics (Inst); Macrogenics (Inst); MedImmune (Inst); Newlink Genetics (Inst); Novartis (Inst); Roche (Inst); Takeda (Inst); Trovagene (Inst) |
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Consulting or Advisory Role - Abbvie; AstraZeneca; Bristol-Myers Squibb; Genentech; Janssen; Lilly; Merck; Xcovery |
Research Funding - Boehringer Ingelheim (Inst); Xcovery (Inst); Xcovery (Inst) |
Other Relationship - Boehringer Ingelheim; Bristol-Myers Squibb |
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Consulting or Advisory Role - Abbvie; ARIAD/Takeda; AstraZeneca; Boehringer Ingelheim; Guardant Health; Novartis; Superdimension |
Research Funding - ARIAD/Takeda (Inst); Guardant Health (Inst); Novartis (Inst) |
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Consulting or Advisory Role - AstraZeneca |
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Consulting or Advisory Role - ARIAD/Takeda; AstraZeneca; Boehringer Ingelheim; Lilly |
Research Funding - ARIAD/Takeda; ArQule; Boehringer Ingelheim; Exelixis; Genentech/Roche; Merck; Nektar; Novartis |
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Stock and Other Ownership Interests - Takeda |
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No Relationships to Disclose |
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Stock and Other Ownership Interests - ARIAD |
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Stock and Other Ownership Interests - ARIAD |
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Stock and Other Ownership Interests - Gatekeeper Pharmaceuticals |
Consulting or Advisory Role - Araxes Pharma; ARIAD; AstraZeneca; Boehringer Ingelheim; Chugai Pharma; Ignyta; Lilly; LOXO; Merrimack; Mirati Therapeutics; Pfizer; Roche/Genentech |
Research Funding - Astellas Pharma; AstraZeneca; Boehringer Ingelheim; Daiichi Sankyo; Lilly; Puma Biotechnology |
Patents, Royalties, Other Intellectual Property - I am a co-inventor on a DFCI owned patent on EGFR mutations licensed to Lab Corp. I receive post-marketing royalties from this invention |